Novel stereocontrolled syntheses of tashiromine and epitashiromine

Scholarly Works

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• Kiss, L.; Semghouli, A.; Remete, A. M.; Novák, T. T. Stereocontrolled Synthesis of Some Novel Azaheterocyclic β-Amino Ester Stereoisomers with Multiple Stereogenic Centers. Synlett 2022, 33, 1655–1659. doi:10.1055/a-1877-3822
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• Kiss, L.; Benke, Z.; Remete, A. M.; Fülöp, F. Diversity-oriented Functionalization of Cyclodienes Through Selective Cycloaddition/Ring-opening/Cross-metathesis Protocols; Transformation of a "Flatland" into Three-dimensional Scaffolds With Stereo- and Regiocontrol. Chemical record (New York, N.Y.) 2020, 20, 1129–1141. doi:10.1002/tcr.202000070
• Kiss, L.; Ouchakour, L.; Abrahami, R. A.; Nonn, M. Stereocontrolled Synthesis of Functionalized Azaheterocycles from Carbocycles through Oxidative Ring Opening/Reductive Ring Closing Protocols. Chemical record (New York, N.Y.) 2019, 20, 120–141. doi:10.1002/tcr.201900025
• Scaggs, W. R.; Scaggs, T. D.; Snaddon, T. N. An enantioselective synthesis of α-alkylated pyrroles via cooperative isothiourea/palladium catalysis. Organic & biomolecular chemistry 2019, 17, 1787–1790. doi:10.1039/c8ob02600a
• Riley, D. L.; Michael, J. P.; de Koning, C. B. New syntheses of (±)-tashiromine and (±)-epitashiromine via enaminone intermediates. Beilstein journal of organic chemistry 2016, 12, 2609–2613. doi:10.3762/bjoc.12.256
• Abrahami, R. A.; Kiss, L.; Barrio, P.; Fülöp, F. Synthesis of fluorinated piperidine and azepane β-amino acid derivatives. Tetrahedron 2016, 72, 7526–7535. doi:10.1016/j.tet.2016.10.005
• Kardos, M.; Kiss, L.; Fülöp, F. Stereocontrolled Synthesis of Difunctionalized Azetidinones and β2, 3-Amino Acid Derivatives from Cyclodienes by Ring-Opening and Cross-Metathesis Reactions. Asian Journal of Organic Chemistry 2015, 4, 1155–1159. doi:10.1002/ajoc.201500286
• Kiss, L.; Forro, E.; Fueloep, F. Novel Stereocontrolled Syntheses of Tashiromine (IV) and Epitashiromine (V). ChemInform 2015, 46. doi:10.1002/chin.201527252

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