Synthesis of carbohydrate-scaffolded thymine glycoconjugates to organize multivalency

Anna K. Ciuk and Thisbe K. Lindhorst
Beilstein J. Org. Chem. 2015, 11, 668–674. https://doi.org/10.3762/bjoc.11.75

Supporting Information

Supporting Information File 1: Experimental and analytical details and NMR spectra for all new synthetic compounds as well as discussion of [2 + 2] photocycloaddition with 7 and 13.
Format: PDF Size: 1.8 MB Download

Cite the Following Article

Synthesis of carbohydrate-scaffolded thymine glycoconjugates to organize multivalency
Anna K. Ciuk and Thisbe K. Lindhorst
Beilstein J. Org. Chem. 2015, 11, 668–674. https://doi.org/10.3762/bjoc.11.75

How to Cite

Ciuk, A. K.; Lindhorst, T. K. Beilstein J. Org. Chem. 2015, 11, 668–674. doi:10.3762/bjoc.11.75

Download Citation

Citation data can be downloaded as file using the "Download" button or used for copy/paste from the text window below.
Citation data in RIS format can be imported by all major citation management software, including EndNote, ProCite, RefWorks, and Zotero.

Citations to This Article

Up to 20 of the most recent references are displayed here.

Scholarly Works

  • Uspenskaia, A.; Doroshenko, I. A.; Popovicheva, K. A.; SHmychkov, N. V.; Pryakhina, E. V.; SHafikov, R. R.; Skvortsov, D. A.; Beklemishev, M. K.; Podrugina, T. A.; Machulkin, A. E.; Beloglazkina, E. K. Pentamethine Cyanine Dyes with Alkynyl Group as Perspective Structure for Conjugation with Targeting Moiety. Elsevier BV 2024. doi:10.2139/ssrn.4897969
  • Uspenskaia, A. A.; Krasnikov, P. A.; Majouga, A. G.; Beloglazkina, E. K.; Machulkin, A. E. Fluorescent conjugates based on prostatic specific membrane antigen ligands as an effective visualization tool for prostate cancer. Биохимия 2023, 88, 1173–1190. doi:10.31857/s0320972523070084
  • Uspenskaia, A. A.; Krasnikov, P. A.; Majouga, A. G.; Beloglazkina, E. K.; Machulkin, A. E. Fluorescent Conjugates Based on Prostate-Specific Membrane Antigen Ligands as an Effective Visualization Tool for Prostate Cancer. Biochemistry. Biokhimiia 2023, 88, 953–967. doi:10.1134/s0006297923070088
  • Machulkin, A. E.; Uspenskaya, A. A.; Zyk, N. Y.; Nimenko, E. A.; Ber, A. P.; Petrov, S. A.; Shafikov, R. R.; Skvortsov, D. A.; Smirnova, G. B.; Borisova, Y. A.; Pokrovsky, V. S.; Kolmogorov, V.; Vaneev, A.; Ivanenkov, Y. A.; Khudyakov, A. D.; Kovalev, S. V.; Erofeev, A.; Gorelkin, P. V.; Beloglazkina, E. K.; Zyk, N. V.; Khazanova, E. S.; Majouga, A. G. PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation. European journal of medicinal chemistry 2021, 227, 113936. doi:10.1016/j.ejmech.2021.113936
  • Jaeschke, S. O.; vom Sondern, I.; Lindhorst, T. K. Synthesis of regioisomeric maltose-based Man/Glc glycoclusters to control glycoligand presentation in 3D space. Organic & biomolecular chemistry 2021, 19, 7013–7023. doi:10.1039/d1ob01150b
  • Brekalo, J.; Despras, G.; Lindhorst, T. K. Pseudoenantiomeric glycoclusters: Synthesis and testing of heterobivalency in carbohydrate-protein interactions. Organic & biomolecular chemistry 2019, 17, 5929–5942. doi:10.1039/c9ob00124g
  • Ciuk, A. K.; Gloe, T.-E.; Lindhorst, T. K. Carbohydrate-Scaffolded Thymine Multimers: Scope and Limitations of the Allylation–Hydroboration Sequence. European Journal of Organic Chemistry 2018, 2018, 6971–6982. doi:10.1002/ejoc.201801387
  • Freichel, T.; Eierhoff, S.; Snyder, N. L.; Hartmann, L. Toward Orthogonal Preparation of Sequence-Defined Monodisperse Heteromultivalent Glycomacromolecules on Solid Support Using Staudinger Ligation and Copper-Catalyzed Click Reactions. The Journal of organic chemistry 2017, 82, 9400–9409. doi:10.1021/acs.joc.7b01398
  • Müller, C.; Despras, G.; Lindhorst, T. K. Organizing multivalency in carbohydrate recognition. Chemical Society reviews 2016, 45, 3275–3302. doi:10.1039/c6cs00165c
  • Poplata, S.; Tröster, A.; Zou, Y.-Q.; Bach, T. Recent Advances in the Synthesis of Cyclobutanes by Olefin [2+2] Photocycloaddition Reactions. Chemical reviews 2016, 116, 9748–9815. doi:10.1021/acs.chemrev.5b00723
  • Haag, R. Multivalency as a chemical organization and action principle. Beilstein journal of organic chemistry 2015, 11, 848–849. doi:10.3762/bjoc.11.94
Other Beilstein-Institut Open Science Activities