Antibacterial structure–activity relationship studies of several tricyclic sulfur-containing flavonoids

Scholarly Works

• Correia, P.; Araújo, P.; Plácido, A.; Pereira, A. R.; Bessa, L. J.; Mateus, N.; de Freitas, V.; Oliveira, J.; Fernandes, I. Light-activated amino-substituted dyes as dual-action antibacterial agents: Bio-efficacy and AFM evaluation. Dyes and Pigments 2024, 224, 111975. doi:10.1016/j.dyepig.2024.111975
• Gosav, S.; Praisler, M.; Cristea, N. P.; Gosav, T.; Paraschiv, C. Experimental and computational studies of 3-(N-morpholinylcarbodithioate)-2-(4-methoxyphenyl)chroman-4-one, a flavanone with potential therapeutical properties. Journal of Molecular Structure 2024, 1295, 136627. doi:10.1016/j.molstruc.2023.136627
• Faleye, O. S.; Boya, B. R.; Lee, J.-H.; Choi, I.; Lee, J. Halogenated Antimicrobial Agents to Combat Drug-Resistant Pathogens. Pharmacological reviews 2023, 76, 90–141. doi:10.1124/pharmrev.123.000863
• Waziri, I.; Kelani, M. T.; Oyedeji-Amusa, M. O.; Oyebamiji, A. K.; Coetzee, L.-C. C.; Adeyinka, A. S.; Muller, A. J. Synthesis and computational investigation of N,N-dimethyl-4-[(Z)-(phenylimino)methyl]aniline derivatives: Biological and quantitative structural activity relationship studies. Journal of Molecular Structure 2023, 1276, 134756. doi:10.1016/j.molstruc.2022.134756
• Thebti, A.; Meddeb, A.; Ben Salem, I.; Bakary, C.; Ayari, S.; Rezgui, F.; Essafi-Benkhadir, K.; Boudabous, A.; Ouzari, H.-I. Antimicrobial Activities and Mode of Flavonoid Actions. Antibiotics (Basel, Switzerland) 2023, 12, 225. doi:10.3390/antibiotics12020225
• Correia, P.; Araújo, P.; Plácido, A.; Pereira, A. R.; Bessa, L. J.; Mateus, N.; de Freitas, V.; Oliveira, J.; Fernandes, I. Light-Activated Amino-Substituted Dyes as Dual-Action Antibacterial Agents: Bio-Efficacy and Afm Evaluation. Elsevier BV 2023. doi:10.2139/ssrn.4648201
• Birsa, M. L.; Sarbu, L. G. An Improved Synthetic Method for Sensitive Iodine Containing Tricyclic Flavonoids. Molecules (Basel, Switzerland) 2022, 27, 8430. doi:10.3390/molecules27238430
• Keekan, K. K.; Ranadive, K. R.; Naik, P.; Sendker, J.; Padmaraj, S. R. Anti-Methicillin-Resistant S. aureus Activity of Fruiting Body and Mycelial Culture Extracts of Xylaria longipes Nitschke (Ascomycota). Pharmaceutical Chemistry Journal 2022, 56, 958–965. doi:10.1007/s11094-022-02733-9
• Moldovan, C.-V.; Savu, M.; Dussert, E.; Aboubacar, H.; Sarbu, L. G.; Matiut, S.; Cudennec, B.; Krier, F.; Ravallec, R.; Birsa, L. M.; Stefan, M. Synthetic Flavonoid BrCl-Flav-An Alternative Solution to Combat ESKAPE Pathogens. Antibiotics (Basel, Switzerland) 2022, 11, 1389. doi:10.3390/antibiotics11101389
• Khadiya, N. M.; Modhavadiya, V. A. CuAAC-Ensembled 1,2,3-Triazole-Linked Biphenyl and N-Arylamide Systems as Diverse Antimicrobial Agents. Russian Journal of Organic Chemistry 2022, 58, 1058–1063. doi:10.1134/s107042802207017x
• Shamsudin, N. F.; Ahmed, Q. U.; Mahmood, S.; Ali Shah, S. A.; Khatib, A.; Mukhtar, S.; Alsharif, M. A.; Parveen, H.; Zakaria, Z. A. Antibacterial Effects of Flavonoids and Their Structure-Activity Relationship Study: A Comparative Interpretation. Molecules (Basel, Switzerland) 2022, 27, 1149. doi:10.3390/molecules27041149
• Fayeulle, A.; Trudel, E.; Damiens, A.; Josse, A.; Youssef, N. B. H.; Vigneron, P.; Vayssade, M.; Rossi, C.; Ceballos, C. Antimicrobial and antioxidant activities of amines derived from vanillin as potential preservatives: Impact of the substituent chain length and polarity. Sustainable Chemistry and Pharmacy 2021, 22, 100471. doi:10.1016/j.scp.2021.100471
• Shao, S.-Y.; Ting, Y.; Wang, J.; Sun, J.; Guo, X.-F. Characterization and identification of the major flavonoids in Phyllostachys edulis leaf extract by UPLC–QTOF–MS/MS. Acta Chromatographica 2020, 32, 228–237. doi:10.1556/1326.2019.00688
• Bahrin, L. G.; Hopf, H.; Jones, P. G.; Birsa, M. L.; Sarbu, L. G. An Approach to Paracyclophane-Based Tetrathiafulvalenes: Synthesis and Characterization of a Pseudo-Geminal [2.2]Paracyclophane 1,3-Dithia-2-Thione. Molecules (Basel, Switzerland) 2020, 25, 5262. doi:10.3390/molecules25225262
• Havasi, M. H.; Ressler, A. J.; Parks, E. L.; Cocolas, A. H.; Weaver, A.; Seeram, N. P.; Henry, G. E. Antioxidant and tyrosinase docking studies of heterocyclic sulfide derivatives containing a thymol moiety. Inorganica Chimica Acta 2020, 505, 119495. doi:10.1016/j.ica.2020.119495
• Sarbu, L. G.; Shova, S.; Peptanariu, D.; Sandu, I. A.; Birsa, L. M.; Bahrin, L. G. The Cytotoxic Properties of Some Tricyclic 1,3-Dithiolium Flavonoids. Molecules (Basel, Switzerland) 2019, 24, 2459. doi:10.3390/molecules24132459
• Sarbu, L. G.; Bahrin, L. G.; Babii, C.; Stefan, M.; Birsa, M. L. Synthetic flavonoids with antimicrobial activity: a review. Journal of applied microbiology 2019, 127, 1282–1290. doi:10.1111/jam.14271
• Sardarian, A. R.; Inaloo, I. D.; Modarresi-Alam, A. R. Highly efficient synthesis of alkyl and aryl primary thiocarbamates and dithiocarbamates under metal- and solvent-free conditions. Molecular diversity 2018, 22, 863–878. doi:10.1007/s11030-018-9831-6
• Ombiro, G. S. o.; Sawai, T.; Noutoshi, Y.; Nishina, Y.; Matsui, H.; Yamamoto, M.; Toyoda, K.; Ichinose, Y. Specific growth inhibitors of Ralstonia solanacearum, Xanthomonas oryzae pv. oryzae, X. campestris pv. campestris, and Clavibacter michiganensis subsp. michiganensis. Microbiological research 2018, 215, 29–35. doi:10.1016/j.micres.2018.06.005
• Sandu, M.; Birsa, L. M.; Bahrin, L. G. Flavonoids – Small Molecules, High Hopes. Acta Chemica Iasi 2017, 25, 6–23. doi:10.1515/achi-2017-0003

Explore citations to this article at