Supporting Information
Supporting Information File 1: Experimental procedures for compounds 5–13, their 1H, 13C NMR, MS, elemental analysis data and the copies of their 1H and 13C NMR spectra. | ||
Format: PDF | Size: 1.2 MB | Download |
Cite the Following Article
The first Pd-catalyzed Buchwald–Hartwig aminations at C-2 or C-4 in the estrone series
Ildikó Bacsa, Dávid Szemerédi, János Wölfling, Gyula Schneider, Lilla Fekete and Erzsébet Mernyák
Beilstein J. Org. Chem. 2018, 14, 998–1003.
https://doi.org/10.3762/bjoc.14.85
How to Cite
Bacsa, I.; Szemerédi, D.; Wölfling, J.; Schneider, G.; Fekete, L.; Mernyák, E. Beilstein J. Org. Chem. 2018, 14, 998–1003. doi:10.3762/bjoc.14.85
Download Citation
Citation data can be downloaded as file using the "Download" button or used for copy/paste from the text window
below.
Citation data in RIS format can be imported by all major citation management software, including EndNote,
ProCite, RefWorks, and Zotero.
Presentation Graphic
Picture with graphical abstract, title and authors for social media postings and presentations. | ||
Format: PNG | Size: 140.6 KB | Download |
Citations to This Article
Up to 20 of the most recent references are displayed here.
Scholarly Works
- Ansari, T. N.; Xu, G.; Preston, A.; Gao, P. Recent Highlights in Micellar Catalysis: An Industrial Outlook. Organic Process Research & Development 2024, 28, 816–830. doi:10.1021/acs.oprd.3c00453
- Firsan, S. J.; Sivakumar, V.; Colacot, T. J. Emerging Trends in Cross-Coupling: Twelve-Electron-Based L1Pd(0) Catalysts, Their Mechanism of Action, and Selected Applications. Chemical reviews 2022, 122, 16983–17027. doi:10.1021/acs.chemrev.2c00204
- Heravi, M. M.; Zadsirjan, V.; Malmir, M.; Mohammadi, L. Buchwald–Hartwig reaction: an update. Monatshefte für Chemie - Chemical Monthly 2021, 152, 1127–1171. doi:10.1007/s00706-021-02834-3
- Kovács, F.; Gopisetty, M. K.; Adamecz, D. I.; Kiricsi, M.; Enyedy, É. A.; Frank, É. Synthesis and conversion of primary and secondary 2-aminoestradiols into A-ring-integrated benzoxazolone hybrids and their in vitro anticancer activity. RSC advances 2021, 11, 13885–13896. doi:10.1039/d1ra01889b
- Traj, P.; Abdolkhaliq, A. H.; Németh, A.; Dajcs, S. T.; Tömösi, F.; Lanisnik-Rizner, T.; Zupkó, I.; Mernyák, E. Transition metal-catalysed A-ring C–H activations and C(sp2)–C(sp2) couplings in the 13α-oestrone series and in vitro evaluation of antiproliferative properties. Journal of enzyme inhibition and medicinal chemistry 2021, 36, 895–902. doi:10.1080/14756366.2021.1900165
- Molnár, Á. Microwave-assisted CN formation reactions. Green Sustainable Process for Chemical and Environmental Engineering and Science; Elsevier, 2021; pp 51–203. doi:10.1016/b978-0-12-819848-3.00002-5
- Zhang, Y.; Takale, B. S.; Gallou, F.; Reilly, J.; Lipshutz, B. H. Sustainable ppm level palladium-catalyzed aminations in nanoreactors under mild, aqueous conditions. Chemical science 2019, 10, 10556–10561. doi:10.1039/c9sc03710a
- Jójárt, R.; Pécsy, S.; Keglevich, G.; Szécsi, M.; Rigó, R.; Özvegy-Laczka, C.; Kecskeméti, G.; Mernyák, E. Pd-Catalyzed microwave-assisted synthesis of phosphonated 13α-estrones as potential OATP2B1, 17β-HSD1 and/or STS inhibitors. Beilstein journal of organic chemistry 2018, 14, 2838–2845. doi:10.3762/bjoc.14.262