Functionalization of the imidazo[1,2-a]pyridine ring in α-phosphonoacrylates and α-phosphonopropionates via microwave-assisted Mizoroki–Heck reaction

Damian Kusy, Agata Wojciechowska, Joanna Małolepsza and Katarzyna M. Błażewska
Beilstein J. Org. Chem. 2020, 16, 15–21. https://doi.org/10.3762/bjoc.16.3

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Functionalization of the imidazo[1,2-a]pyridine ring in α-phosphonoacrylates and α-phosphonopropionates via microwave-assisted Mizoroki–Heck reaction
Damian Kusy, Agata Wojciechowska, Joanna Małolepsza and Katarzyna M. Błażewska
Beilstein J. Org. Chem. 2020, 16, 15–21. https://doi.org/10.3762/bjoc.16.3

How to Cite

Kusy, D.; Wojciechowska, A.; Małolepsza, J.; Błażewska, K. M. Beilstein J. Org. Chem. 2020, 16, 15–21. doi:10.3762/bjoc.16.3

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  • Tali, J. A.; Kumar, G.; Sharma, B. K.; Rasool, Y.; Sharma, Y.; Shankar, R. Synthesis and site selective C-H functionalization of imidazo-[1,2-a]pyridines. Organic & biomolecular chemistry 2023, 21, 7267–7289. doi:10.1039/d3ob00849e
  • Małolepsza, J.; Marchwicka, A.; Serwa, R. A.; Niinivehmas, S. P.; Pentikäinen, O. T.; Gendaszewska-Darmach, E.; Błażewska, K. M. Rational design, optimization, and biological evaluation of novel α-Phosphonopropionic acids as covalent inhibitors of Rab geranylgeranyl transferase. Journal of enzyme inhibition and medicinal chemistry 2022, 37, 940–951. doi:10.1080/14756366.2022.2053525
  • Kusy, D.; Marchwicka, A.; Małolepsza, J.; Justyna, K.; Gendaszewska-Darmach, E.; Błażewska, K. M. Synthesis of the 6-Substituted Imidazo[1,2-a]Pyridine-3-yl-2- Phosphonopropionic Acids as Potential Inhibitors of Rab Geranylgeranyl Transferase. Frontiers in chemistry 2021, 8, 596162. doi:10.3389/fchem.2020.596162
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