Novel library synthesis of 3,4-disubstituted pyridin-2(1H)-ones via cleavage of pyridine-2-oxy-7-azabenzotriazole ethers under ionic hydrogenation conditions at room temperature

Romain Pierre, Anne Brethon, Sylvain A. Jacques, Aurélie Blond, Sandrine Chambon, Sandrine Talano, Catherine Raffin, Branislav Musicki, Claire Bouix-Peter, Loic Tomas, Gilles Ouvry, Rémy Morgentin, Laurent F. Hennequin and Craig S. Harris
Beilstein J. Org. Chem. 2021, 17, 156–165. https://doi.org/10.3762/bjoc.17.16

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Novel library synthesis of 3,4-disubstituted pyridin-2(1H)-ones via cleavage of pyridine-2-oxy-7-azabenzotriazole ethers under ionic hydrogenation conditions at room temperature
Romain Pierre, Anne Brethon, Sylvain A. Jacques, Aurélie Blond, Sandrine Chambon, Sandrine Talano, Catherine Raffin, Branislav Musicki, Claire Bouix-Peter, Loic Tomas, Gilles Ouvry, Rémy Morgentin, Laurent F. Hennequin and Craig S. Harris
Beilstein J. Org. Chem. 2021, 17, 156–165. https://doi.org/10.3762/bjoc.17.16

How to Cite

Pierre, R.; Brethon, A.; Jacques, S. A.; Blond, A.; Chambon, S.; Talano, S.; Raffin, C.; Musicki, B.; Bouix-Peter, C.; Tomas, L.; Ouvry, G.; Morgentin, R.; Hennequin, L. F.; Harris, C. S. Beilstein J. Org. Chem. 2021, 17, 156–165. doi:10.3762/bjoc.17.16

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  • PRYDE DAVID CAMERON; SHRIVASTAVA RITESH KUMAR; YADAV DHARMENDRA B; GHOSH RAJIB; BASU SOURAV; BANERJEE MONALI; MIDDYA SANDIP KUMAR; DEBNATH SABYASACHI; SURYA ARJUN. PYRIDONE AND PYRIMIDINONE INHIBITORS OF HEMATOPOIETIC PROGENITOR KINASE 1. WO 2024105363 A1, May 23, 2024.
  • BANERJEE MONALI; SHRIVASTAVA RITESH KUMAR; MIDDYA SANDIP KUMAR; DEBNATH SABYASACHI; PRYDE DAVID CAMERON; BASU SOURAV; GHOSH RAJIB; YADAV DHARMENDRA B; SURYA ARJUN. HETEROCYCLIC INHIBITORS OF CDC-LIKE KINASES. WO 2024105364 A1, May 23, 2024.
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