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Search for "Michael additions" in Full Text gives 51 result(s) in Beilstein Journal of Organic Chemistry.

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Amines as key building blocks in Pd-assisted multicomponent processes

Didier Bouyssi,
Nuno Monteiro and
Geneviève Balme

Beilstein J. Org. Chem. 2011, 7, 1387–1406, doi:10.3762/bjoc.7.163

transformations, including aza-Michael additions, hydroaminations of alkynes, Buchwald–Hartwig aminations, and allylic aminations, thereby allowing the creation of several covalent bonds in a single operation. Imine derivatives are also of high synthetic value as they may act either as electrophilic or

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Graphical Abstract

Scheme 1: Synthesis of substituted amides.

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Scheme 2: Synthesis of ketocarbamates and imidazolones.

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Scheme 3: Access to β-lactams.

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Scheme 4: Access to β-lactams with increased structural diversity.

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Scheme 5: Synthesis of imidazolinium salts.

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Scheme 6: Access to the indenamine core.

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Scheme 7: Synthesis of substituted tetrahydropyridines.

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Scheme 8: Synthesis of more substituted tetrahydropyridines.

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Scheme 9: Synthesis of chiral tetrahydropyridines.

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Scheme 10: Preparation of α-aminonitrile by a catalyzed Strecker reaction.

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Scheme 11: Synthesis of spiroacetals.

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Scheme 12: Synthesis of masked 3-aminoindan-1-ones.

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Scheme 13: Synthesis of homoallylic amines and α-aminoesters.

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Scheme 14: Preparation of 1,2-dihydroisoquinolin-1-ylphosphonates.

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Scheme 15: Pyrazole elaboration by cycloaddition of hydrazines with alkynones generated in situ.

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Scheme 16: An alternative approach to pyrazoles involving hydrazine cycloaddition.

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Scheme 17: Synthesis of pyrroles by cyclization of propargyl amines.

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Scheme 18: Isoindolone and phthalazone synthesis by cyclization of acylhydrazides.

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Scheme 19: Sultam synthesis by cyclization of sulfonamides.

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Scheme 20: Synthesis of sulfonamides by aminosulfonylation of aryl iodides.

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Scheme 21: Pyrrolidine synthesis by carbopalladation of allylamines.

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Scheme 22: Synthesis of indoles through a sequential C–C coupling/desilylation–coupling/cyclization reaction.

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Scheme 23: Synthesis of indoles by a site selective Pd/C catalyzed cross-coupling approach.

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Scheme 24: Synthesis of isoindolin-1-one derivatives through a sequential Sonogashira coupling/carbonylation/h...

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Scheme 25: Synthesis of pyrroles through an allylic amination/Sonogashira coupling/hydroamination reaction.

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Scheme 26: Synthesis of indoles through a Sonogashira coupling/cyclofunctionalization reaction.

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Scheme 27: Synthesis of indoles through a one-pot two-step Sonogashira coupling/cyclofunctionalization reactio...

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Scheme 28: Synthesis of α-alkynylindoles through a Pd-catalyzed Sonogashira/double C–N coupling reaction.

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Scheme 29: Synthesis of indoles through a Pd-catalyzed sequential alkenyl amination/C-arylation/N-arylation.

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Scheme 30: Synthesis of N-aryl-2-benzylpyrrolidines through a sequential N-arylation/carboamination reaction.

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Scheme 31: Synthesis of phenothiazine derivatives through a one-pot palladium-catalyzed double C–N arylation i...

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Scheme 32: Synthesis of substituted imidazolidinones through a palladium-catalyzed three-component reaction of...

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Scheme 33: Synthesis of 2,3-diarylated amines through a palladium-catalyzed four-component reaction involving ...

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Scheme 34: Synthesis of rolipram involving a Pd-catalyzed three-component reaction.

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Scheme 35: Synthesis of seven-membered ring lactams through a Pd-catalyzed amination/intramolecular cyclocarbo...

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Review

Published 10 Oct 2011

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