Synthesis and biological profile of 2,3-dihydro[1,3]thiazolo[4,5-b]pyridines, a novel class of acyl-ACP thioesterase inhibitors

Jens Frackenpohl, David M. Barber, Guido Bojack, Birgit Bollenbach-Wahl, Ralf Braun, Rahel Getachew, Sabine Hohmann, Kwang-Yoon Ko, Karoline Kurowski, Bernd Laber, Rebecca L. Mattison, Thomas Müller, Anna M. Reingruber, Dirk Schmutzler and Andrea Svejda
Beilstein J. Org. Chem. 2024, 20, 540–551. https://doi.org/10.3762/bjoc.20.46

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Supporting Information File 1: General synthetic procedures, characterization of all target compounds, methods for biological and biochemical testing, and scans of 1H and 13C NMR spectra of the new 2,3-dihydro[1,3]thiazolo[4,5-b]pyridines.
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Synthesis and biological profile of 2,3-dihydro[1,3]thiazolo[4,5-b]pyridines, a novel class of acyl-ACP thioesterase inhibitors
Jens Frackenpohl, David M. Barber, Guido Bojack, Birgit Bollenbach-Wahl, Ralf Braun, Rahel Getachew, Sabine Hohmann, Kwang-Yoon Ko, Karoline Kurowski, Bernd Laber, Rebecca L. Mattison, Thomas Müller, Anna M. Reingruber, Dirk Schmutzler and Andrea Svejda
Beilstein J. Org. Chem. 2024, 20, 540–551. https://doi.org/10.3762/bjoc.20.46

How to Cite

Frackenpohl, J.; Barber, D. M.; Bojack, G.; Bollenbach-Wahl, B.; Braun, R.; Getachew, R.; Hohmann, S.; Ko, K.-Y.; Kurowski, K.; Laber, B.; Mattison, R. L.; Müller, T.; Reingruber, A. M.; Schmutzler, D.; Svejda, A. Beilstein J. Org. Chem. 2024, 20, 540–551. doi:10.3762/bjoc.20.46

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