Synthesis of 1,4-azaphosphinine nucleosides and evaluation as inhibitors of human cytidine deaminase and APOBEC3A

Maksim V. Kvach, Stefan Harjes, Harikrishnan M. Kurup, Geoffrey B. Jameson, Elena Harjes and Vyacheslav V. Filichev
Beilstein J. Org. Chem. 2024, 20, 1088–1098. https://doi.org/10.3762/bjoc.20.96

Supporting Information

Supporting Information File 1: Supplementary experimental details about the enzymatic assays and the synthesis of nucleosides and modified ODNs, assignment of 1H, 13C, 31P NMR and IR spectra and results of HRESIMS experiments for new compounds synthesised as well as RP-HPLC profiles and HRESIMS spectra of ODNs.
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Synthesis of 1,4-azaphosphinine nucleosides and evaluation as inhibitors of human cytidine deaminase and APOBEC3A
Maksim V. Kvach, Stefan Harjes, Harikrishnan M. Kurup, Geoffrey B. Jameson, Elena Harjes and Vyacheslav V. Filichev
Beilstein J. Org. Chem. 2024, 20, 1088–1098. https://doi.org/10.3762/bjoc.20.96

How to Cite

Kvach, M. V.; Harjes, S.; Kurup, H. M.; Jameson, G. B.; Harjes, E.; Filichev, V. V. Beilstein J. Org. Chem. 2024, 20, 1088–1098. doi:10.3762/bjoc.20.96

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