Supporting Information
Supporting Information File 1: Experimental details and characterization data for all compounds. | ||
Format: PDF | Size: 1.5 MB | Download |
Cite the Following Article
An easy direct arylation of 5-pyrazolones
Hao Gong, Yiwen Yang, Zechao Wang and Chunxiang Kuang
Beilstein J. Org. Chem. 2013, 9, 2033–2039.
https://doi.org/10.3762/bjoc.9.240
How to Cite
Gong, H.; Yang, Y.; Wang, Z.; Kuang, C. Beilstein J. Org. Chem. 2013, 9, 2033–2039. doi:10.3762/bjoc.9.240
Download Citation
Citation data can be downloaded as file using the "Download" button or used for copy/paste from the text window
below.
Citation data in RIS format can be imported by all major citation management software, including EndNote,
ProCite, RefWorks, and Zotero.
Citations to This Article
Up to 20 of the most recent references are displayed here.
Scholarly Works
- Kittikool, T.; Viriyanukul, T.; Phakdeeyothin, K.; Yotphan, S. Switchable Site‐Selectivite Direct Acetoxylation of Pyrazolones. Asian Journal of Organic Chemistry 2025. doi:10.1002/ajoc.202400808
- Zheng, T.; Yu, Z.; Li, J.; Gu, Q.; Gu, L.; Li, Z.; Ma, W. Solvent‐Free Dehydrogenative C−H Chalcogenations of Pyrazolones Using Mechanochemistry. Asian Journal of Organic Chemistry 2024, 13. doi:10.1002/ajoc.202400353
- Li, M.; Yang, S.; Zhang, J.; Gao, Z.; Zheng, L.; Lu, F.; Feng, Y. Electrochemical oxidative selective halogenation of pyrazolones for the synthesis of 4-halopyrazolones. Organic & biomolecular chemistry 2024, 22, 6080–6084. doi:10.1039/d4ob00982g
- Matsumura, M.; Nakamura, A.; Yanagida, A.; Murata, Y.; Yasuike, S. Copper-catalyzed three-component reaction of pyrazol-3-ones (antipyrine), triarylbismuthines, and selenium: Synthesis of 4-selanylpyrazol-3-ones. Tetrahedron 2023, 142, 133526. doi:10.1016/j.tet.2023.133526
- Lu, F.; Hu, L.; Zhang, J.; Feng, Y. Electrochemical Oxidative Cross‐Coupling of Pyrazolones and Diselenides to Construct C‐Se Bonds. Asian Journal of Organic Chemistry 2023, 12. doi:10.1002/ajoc.202200719
- Purohit, V. B.; Prajapati, R. V.; Prajapati, V. D.; Karad, S. C.; Sapariya, N. H.; Avalani, J. R.; Raval, D. K. C−H Functionalization Reactions of 1‐Aryl‐5‐pyrazolones. European Journal of Organic Chemistry 2022, 2022. doi:10.1002/ejoc.202201111
- Phakdeeyothin, K.; Viriyanukul, T.; Udomsasporn, K.; Phomphrai, K.; Yotphan, S. Metal‐Free Aminomethylation of Pyrazolones: Direct Access to 4‐Aminomethylated Pyrazolones. Asian Journal of Organic Chemistry 2022, 11. doi:10.1002/ajoc.202200467
- Konishi, K.; Yasui, M.; Miki, K.; Takeda, N.; Ueda, M. Construction of pyrazolodiazepines using AuI, a dual functional gold catalyst. Organic & biomolecular chemistry 2022, 20, 3382–3386. doi:10.1039/d2ob00199c
- Wen, K.; Wu, Y.; Chen, J.; Shi, J.; Zheng, M.; Yao, X.; Tang, X. Copper-Mediated Decarboxylative Coupling of 3-Indoleacetic Acids with Pyrazolones. ACS omega 2022, 7, 5274–5282. doi:10.1021/acsomega.1c06443
- Dong, C.; Xiangzhen, M.; Wang, D.; Zhao, X.; Yusheng, W.; Zhiyu, J. A palladium-catalyzed cascade approach for the synthesis of 3,3a,4,6,7,8,9,9a-octahydro-1H-benzo[f]isoindole-1,5(2H)-diones. Journal of Chemical Research 2021, 45, 174751982110586–1113. doi:10.1177/17475198211058653
- Shchegolkov, E. V.; Burgart, Y. V.; Matsneva, D. A.; Borisevich, S. S.; Kadyrova, R. A.; Orshanskaya, I. R.; Zarubaev, V. V.; Saloutin, V. I. Polyfluoroalkylated antipyrines in Pd-catalyzed transformations. RSC advances 2021, 11, 35174–35181. doi:10.1039/d1ra06967e
- Sonowal, P.; Bhorali, P.; Sultana, S.; Gogoi, S. Pd(ii)-Catalyzed regioselective functionalization of antipyrines: synthesis of pyrazolono-maleimides and pyrazolono-quinones. Organic & biomolecular chemistry 2021, 19, 5333–5341. doi:10.1039/d1ob00819f
- Akhmadiev, N. S.; Mescheryakova, E. S.; Akhmetova, V. R.; Khairullina, V. R.; Khalilov, L. M.; Ibragimov, A. G. Synthesis, Crystal Structure and Docking Studies as Potential Anti-Inflammatory Agents of Novel Antipyrine Sulfanyl Derivatives. Journal of Molecular Structure 2021, 1228, 129734. doi:10.1016/j.molstruc.2020.129734
- Sasmal, A.; Bera, J. K.; Doucet, H.; Soulé, J.-F. Reactivity of antipyrine and haloantipyrines in Pd-catalyzed CH bond arylations. Tetrahedron Letters 2020, 61, 151798. doi:10.1016/j.tetlet.2020.151798
- Kittikool, T.; Yotphan, S. Metal‐Free Direct C−H Thiolation and Thiocyanation of Pyrazolones. European Journal of Organic Chemistry 2020, 2020, 961–970. doi:10.1002/ejoc.201901770
- Zhang, Y.; Nie, L.-J.; Luo, L.; Mao, J.-X.; Liu, J.-X.; Xu, G.-H.; Chen, D.; Luo, H.-Q. The selective condensation of pyrazolones to isatins in aqueous medium. Tetrahedron 2020, 76, 130916. doi:10.1016/j.tet.2019.130916
- Kovalev, I. S.; Savchuk, M. I.; Kopchuk, D. S.; Zyryanov, G. V.; Pospelova, T. A.; Rusinov, V. L.; Chupakhin, O. N. A Convenient Synthetic Approach to Phenazone Derivatives Containing a 1,2,4-Triazine or Pyridine Fragment. Russian Journal of Organic Chemistry 2019, 55, 886–889. doi:10.1134/s1070428019060228
- Xiao, Y.; Wu, X.; Teng, J.; Sun, S.; Yu, J.-T.; Cheng, J. Copper-catalyzed acylation of pyrazolones with aldehydes to afford 4-acylpyrazolones. Organic & biomolecular chemistry 2019, 17, 7552–7557. doi:10.1039/c9ob01486a
- Kittikool, T.; Thupyai, A.; Phomphrai, K.; Yotphan, S. Copper/Persulfate-Promoted Oxidative Decarboxylative C−H Acylation of Pyrazolones with α-Oxocarboxylic Acids: Direct Access to 4-Acylpyrazolones under Mild Conditions. Advanced Synthesis & Catalysis 2018, 360, 3345–3355. doi:10.1002/adsc.201800464
- Thupyai, A.; Pimpasri, C.; Yotphan, S. DABCO-catalyzed silver-promoted direct thiolation of pyrazolones with diaryl disulfides. Organic & biomolecular chemistry 2018, 16, 424–432. doi:10.1039/c7ob02860a