Peptide stapling by late-stage Suzuki–Miyaura cross-coupling
- Hendrik Gruß,
- Rebecca C. Feiner,
- Ridhiwan Mseya,
- David C. Schröder,
- Michał Jewgiński,
- Kristian M. Müller,
- Rafał Latajka,
- Antoine Marion and
- Norbert Sewald
Beilstein J. Org. Chem. 2022, 18, 1–12, doi:10.3762/bjoc.18.1
The enzyme mechanism of patchoulol synthase
- Houchao Xu,
- Bernd Goldfuss,
- Gregor Schnakenburg and
- Jeroen S. Dickschat
Beilstein J. Org. Chem. 2022, 18, 13–24, doi:10.3762/bjoc.18.2
Bifunctional thiourea-catalyzed asymmetric [3 + 2] annulation reactions of 2-isothiocyanato-1-indanones with barbiturate-based olefins
- Jiang-Song Zhai and
- Da-Ming Du
Beilstein J. Org. Chem. 2022, 18, 25–36, doi:10.3762/bjoc.18.3
Recent advances and perspectives in ruthenium-catalyzed cyanation reactions
- Thaipparambil Aneeja,
- Cheriya Mukkolakkal Abdulla Afsina,
- Padinjare Veetil Saranya and
- Gopinathan Anilkumar
Beilstein J. Org. Chem. 2022, 18, 37–52, doi:10.3762/bjoc.18.4
1,2-Naphthoquinone-4-sulfonic acid salts in organic synthesis
- Ruan Carlos B. Ribeiro,
- Patricia G. Ferreira,
- Amanda de A. Borges,
- Luana da S. M. Forezi,
- Fernando de Carvalho da Silva and
- Vitor F. Ferreira
Beilstein J. Org. Chem. 2022, 18, 53–69, doi:10.3762/bjoc.18.5
Efficient synthesis of ethyl 2-(oxazolin-2-yl)alkanoates via ethoxycarbonylketene-induced electrophilic ring expansion of aziridines
- Yelong Lei and
- Jiaxi Xu
Beilstein J. Org. Chem. 2022, 18, 70–76, doi:10.3762/bjoc.18.6
Efficient and regioselective synthesis of dihydroxy-substituted 2-aminocyclooctane-1-carboxylic acid and its bicyclic derivatives
- İlknur Polat,
- Selçuk Eşsiz,
- Uğur Bozkaya and
- Emine Salamci
Beilstein J. Org. Chem. 2022, 18, 77–85, doi:10.3762/bjoc.18.7
Earth-abundant 3d transition metals on the rise in catalysis
- Nikolaos Kaplaneris and
- Lutz Ackermann
Beilstein J. Org. Chem. 2022, 18, 86–88, doi:10.3762/bjoc.18.8
Chemoselective N-acylation of indoles using thioesters as acyl source
- Tianri Du,
- Xiangmu Wei,
- Honghong Xu,
- Xin Zhang,
- Ruiru Fang,
- Zheng Yuan,
- Zhi Liang and
- Yahui Li
Beilstein J. Org. Chem. 2022, 18, 89–94, doi:10.3762/bjoc.18.9
Chemical and chemoenzymatic routes to bridged homoarabinofuranosylpyrimidines: Bicyclic AZT analogues
- Sandeep Kumar,
- Jyotirmoy Maity,
- Banty Kumar,
- Sumit Kumar and
- Ashok K. Prasad
Beilstein J. Org. Chem. 2022, 18, 95–101, doi:10.3762/bjoc.18.10
Regioselective synthesis of methyl 5-(N-Boc-cycloaminyl)-1,2-oxazole-4-carboxylates as new amino acid-like building blocks
- Jolita Bruzgulienė,
- Greta Račkauskienė,
- Aurimas Bieliauskas,
- Vaida Milišiūnaitė,
- Miglė Dagilienė,
- Gita Matulevičiūtė,
- Vytas Martynaitis,
- Sonata Krikštolaitytė,
- Frank A. Sløk and
- Algirdas Šačkus
Beilstein J. Org. Chem. 2022, 18, 102–109, doi:10.3762/bjoc.18.11
Tenacibactins K–M, cytotoxic siderophores from a coral-associated gliding bacterium of the genus Tenacibaculum
- Yasuhiro Igarashi,
- Yiwei Ge,
- Tao Zhou,
- Amit Raj Sharma,
- Enjuro Harunari,
- Naoya Oku and
- Agus Trianto
Beilstein J. Org. Chem. 2022, 18, 110–119, doi:10.3762/bjoc.18.12
Mechanistic studies of the solvolysis of alkanesulfonyl and arenesulfonyl halides
- Malcolm J. D’Souza and
- Dennis N. Kevill
Beilstein J. Org. Chem. 2022, 18, 120–132, doi:10.3762/bjoc.18.13
Green synthesis of C5–C6-unsubstituted 1,4-DHP scaffolds using an efficient Ni–chitosan nanocatalyst under ultrasonic conditions
- Soumyadip Basu,
- Sauvik Chatterjee,
- Suman Ray,
- Suvendu Maity,
- Prasanta Ghosh,
- Asim Bhaumik and
- Chhanda Mukhopadhyay
Beilstein J. Org. Chem. 2022, 18, 133–142, doi:10.3762/bjoc.18.14
Ready access to 7,8-dihydroindolo[2,3-d][1]benzazepine-6(5H)-one scaffold and analogues via early-stage Fischer ring-closure reaction
- Irina Kuznetcova,
- Felix Bacher,
- Daniel Vegh,
- Hsiang-Yu Chuang and
- Vladimir B. Arion
Beilstein J. Org. Chem. 2022, 18, 143–151, doi:10.3762/bjoc.18.15
High-speed C–H chlorination of ethylene carbonate using a new photoflow setup
- Takayoshi Kasakado,
- Takahide Fukuyama,
- Tomohiro Nakagawa,
- Shinji Taguchi and
- Ilhyong Ryu
Beilstein J. Org. Chem. 2022, 18, 152–158, doi:10.3762/bjoc.18.16
Synthesis and bioactivity of pyrrole-conjugated phosphopeptides
- Qiuxin Zhang,
- Weiyi Tan and
- Bing Xu
Beilstein J. Org. Chem. 2022, 18, 159–166, doi:10.3762/bjoc.18.17
Asymmetric organocatalytic Michael addition of cyclopentane-1,2-dione to alkylidene oxindole
- Estelle Silm,
- Ivar Järving and
- Tõnis Kanger
Beilstein J. Org. Chem. 2022, 18, 167–173, doi:10.3762/bjoc.18.18
Synthesis and late stage modifications of Cyl derivatives
- Phil Servatius and
- Uli Kazmaier
Beilstein J. Org. Chem. 2022, 18, 174–181, doi:10.3762/bjoc.18.19
Multi-faceted reactivity of N-fluorobenzenesulfonimide (NFSI) under mechanochemical conditions: fluorination, fluorodemethylation, sulfonylation, and amidation reactions
- José G. Hernández,
- Karen J. Ardila-Fierro,
- Dajana Barišić and
- Hervé Geneste
Beilstein J. Org. Chem. 2022, 18, 182–189, doi:10.3762/bjoc.18.20
Diametric calix[6]arene-based phosphine gold(I) cavitands
- Gabriele Giovanardi,
- Andrea Secchi,
- Arturo Arduini and
- Gianpiero Cera
Beilstein J. Org. Chem. 2022, 18, 190–196, doi:10.3762/bjoc.18.21
The role of chemistry in the success of oligonucleotides as therapeutics
- Pawan Kumar and
- Tom Brown
Beilstein J. Org. Chem. 2022, 18, 197–199, doi:10.3762/bjoc.18.22
Glycosylated coumarins, flavonoids, lignans and phenylpropanoids from Wikstroemia nutans and their biological activities
- Meifang Wu,
- Xiangdong Su,
- Yichuang Wu,
- Yuanjing Luo,
- Ying Guo and
- Yongbo Xue
Beilstein J. Org. Chem. 2022, 18, 200–207, doi:10.3762/bjoc.18.23
Anomeric 1,2,3-triazole-linked sialic acid derivatives show selective inhibition towards a bacterial neuraminidase over a trypanosome trans-sialidase
- Peterson de Andrade,
- Sanaz Ahmadipour and
- Robert A. Field
Beilstein J. Org. Chem. 2022, 18, 208–216, doi:10.3762/bjoc.18.24
Organocatalytic asymmetric nitroso aldol reaction of α-substituted malonamates
- Ekta Gupta,
- Narendra Kumar Vaishanv,
- Sandeep Kumar,
- Raja Krishnan Purshottam,
- Ruchir Kant and
- Kishor Mohanan
Beilstein J. Org. Chem. 2022, 18, 217–224, doi:10.3762/bjoc.18.25
Trichloroacetic acid fueled practical amine purifications
- Aleena Thomas,
- Baptiste Gasch,
- Enzo Olivieri and
- Adrien Quintard
Beilstein J. Org. Chem. 2022, 18, 225–231, doi:10.3762/bjoc.18.26
Flow synthesis of oxadiazoles coupled with sequential in-line extraction and chromatography
- Kian Donnelly and
- Marcus Baumann
Beilstein J. Org. Chem. 2022, 18, 232–239, doi:10.3762/bjoc.18.27
New advances in asymmetric organocatalysis
- Radovan Šebesta
Beilstein J. Org. Chem. 2022, 18, 240–242, doi:10.3762/bjoc.18.28
Synthesis of novel [1,2,4]triazolo[1,5-b][1,2,4,5]tetrazines and investigation of their fungistatic activity
- Anna V. Korotina,
- Svetlana G. Tolshchina,
- Rashida I. Ishmetova,
- Natalya P. Evstigneeva,
- Natalya A. Gerasimova,
- Natalya V. Zilberberg,
- Nikolay V. Kungurov,
- Gennady L. Rusinov,
- Oleg N. Chupakhin and
- Valery N. Charushin
Beilstein J. Org. Chem. 2022, 18, 243–250, doi:10.3762/bjoc.18.29
Iridium-catalyzed hydroacylation reactions of C1-substituted oxabenzonorbornadienes with salicylaldehyde: an experimental and computational study
- Angel Ho,
- Austin Pounder,
- Krish Valluru,
- Leanne D. Chen and
- William Tam
Beilstein J. Org. Chem. 2022, 18, 251–261, doi:10.3762/bjoc.18.30
Recent developments and trends in the iron- and cobalt-catalyzed Sonogashira reactions
- Surendran Amrutha,
- Sankaran Radhika and
- Gopinathan Anilkumar
Beilstein J. Org. Chem. 2022, 18, 262–285, doi:10.3762/bjoc.18.31
New efficient synthesis of polysubstituted 3,4-dihydroquinazolines and 4H-3,1-benzothiazines through a Passerini/Staudinger/aza-Wittig/addition/nucleophilic substitution sequence
- Long Zhao,
- Mao-Lin Yang,
- Min Liu and
- Ming-Wu Ding
Beilstein J. Org. Chem. 2022, 18, 286–292, doi:10.3762/bjoc.18.32
Regioselectivity of the SEAr-based cyclizations and SEAr-terminated annulations of 3,5-unsubstituted, 4-substituted indoles
- Jonali Das and
- Sajal Kumar Das
Beilstein J. Org. Chem. 2022, 18, 293–302, doi:10.3762/bjoc.18.33
