Highly selective difluoromethylations of β-keto amides with TMSCF2Br under mild conditions

  • Yakun Wang,
  • Shuaifei Wang,
  • Conghui Zhang,
  • Ting Zhao,
  • Yanqin Hu,
  • Mingwei Zhang,
  • Pengli Chen,
  • Yang Fu and
  • Jieli Lv
Published 20 Apr 2021
Beilstein Arch. 2021, 202135. doi:10.3762/bxiv.2021.35.v1
Published 14 Apr 2021
Beilstein Arch. 2021, 202133. doi:10.3762/bxiv.2021.33.v1
Published 06 Apr 2021
Beilstein Arch. 2021, 202131. doi:10.3762/bxiv.2021.31.v1
Published 23 Mar 2021
Beilstein Arch. 2021, 202128. doi:10.3762/bxiv.2021.28.v1

Me3Al mediated domino nucleophilic addition/intramolecular cyclisation of 2-(2-oxo-2-phenylethyl)benzonitriles with amines; A convenient approach for the synthesis of substituted 1-aminoisoquinolines

  • Midhun Sai Krishna Adusumalli,
  • Lakshmi Narayana Sharma Konidena,
  • Hima Bindu Gandham,
  • Krishnaiah Kumari,
  • Krishna Reddy Valluru,
  • Satya Kameswara Rao Nidasanametla,
  • Venkateswara Rao Battula and
  • Hari Krishna Namballa
Published 22 Mar 2021
Beilstein Arch. 2021, 202126. doi:10.3762/bxiv.2021.26.v1
Published 22 Mar 2021
Beilstein Arch. 2021, 202125. doi:10.3762/bxiv.2021.25.v1
Published 15 Mar 2021
Beilstein Arch. 2021, 202122. doi:10.3762/bxiv.2021.22.v1

Structural Effects of meso-Halogenation on Porphyrins: meso-Xn-ABCD Macrocycles

  • Keith J. Flanagan,
  • Maximilian Paradiz Dominguez,
  • Zoi Melissari,
  • Hans-Georg Eckhardt,
  • René M. Williams,
  • Dáire Gibbons,
  • Caroline Prior,
  • Gemma M. Locke,
  • Alina Meindl,
  • Aoife A. Ryan and
  • Mathias O Senge
Published 12 Mar 2021
Beilstein Arch. 2021, 202121. doi:10.3762/bxiv.2021.21.v1

Synthesis and transformation of sphingosine analogue pinane-based 2-amino-1,3-diols

  • Ákos Bajtel,
  • Mounir Raji,
  • Matti Haukka,
  • Ferenc Fülöp and
  • Zsolt Szakonyi
Published 11 Mar 2021
Beilstein Arch. 2021, 202120. doi:10.3762/bxiv.2021.20.v1

Synthesis of bis-aryloxyfluoromethanes

  • Carl Recsei and
  • Yaniv Barda
Published 09 Mar 2021
Beilstein Arch. 2021, 202119. doi:10.3762/bxiv.2021.19.v1

DBU-catalyzed Michael addition of bulky glycine imine to α,β-unsaturated isoxazoles and pyrazolamides

  • Yu-Jun Bai,
  • Mei-Ling Cheng,
  • Xiao-Mu Hu,
  • Ya-Jun Bai,
  • Xiao-Hui Zheng,
  • Sheng-Yong Zhang and
  • Ping-An Wang
Published 09 Mar 2021
Beilstein Arch. 2021, 202118. doi:10.3762/bxiv.2021.18.v1
Published 08 Mar 2021
Beilstein Arch. 2021, 202117. doi:10.3762/bxiv.2021.17.v1

Substituted Nitrogen-Bridged Diazocines

  • Pascal Lentes,
  • Jeremy Rudtke and
  • Rainer Herges
Published 08 Mar 2021
Beilstein Arch. 2021, 202116. doi:10.3762/bxiv.2021.16.v1

Blue Light induced Coupling of N-Hydroxysulphonamides: An efficient and green Approach to Access Symmetrical Thiosulfonates

  • Arvind Kumar Pandey,
  • Akhilesh Kumar,
  • Narsingh Verma and
  • Santosh Kumar Srivastava
Published 05 Mar 2021
Beilstein Arch. 2021, 202115. doi:10.3762/bxiv.2021.15.v1
Published 25 Feb 2021
Beilstein Arch. 2021, 202114. doi:10.3762/bxiv.2021.14.v1

Computational model predicts protein binding sites of a luminescent ligand equipped with guanidiniocarbonyl-pyrrole groups

  • Neda Rafieiolhosseini,
  • Matthias Killa,
  • Niklas Tötsch,
  • Jean-Noël Grad,
  • Alexander Höing,
  • Christian Ottmann,
  • Shirley K. Knauer,
  • Jens Voskuhl and
  • Daniel Hoffmann
Published 19 Feb 2021
Beilstein Arch. 2021, 202111. doi:10.3762/bxiv.2021.11.v1

Synthesis of multiply fluorinated N-acetyl-D-glucosamine and D-galactosamine analogs via the corresponding deoxyfluorinated glucosazide and galactosazide thiodonors

  • Vojtěch Hamala,
  • Lucie Červenková Šťastná,
  • Martin Kurfiřt,
  • Petra Cuřínová,
  • Martin Dračínský and
  • Jindřich Karban
Published 11 Feb 2021
Beilstein Arch. 2021, 202110. doi:10.3762/bxiv.2021.10.v1

Enhanced cell target specificity and uptake of lipid nanoparticles using RNA aptamers and peptides

  • Roslyn M. Ray,
  • Anders Højgaard Hansen,
  • Maria Taskova,
  • Bernhard Jandl,
  • Jonas Hansen,
  • Citra Soemardy,
  • Kevin V. Morris and
  • Kira Astakhova
Published 26 Jan 2021
Beilstein Arch. 2021, 20217. doi:10.3762/bxiv.2021.7.v1

Total Synthesis of Pyrrolo[2,3-c]quinoline Alkaloid: Trigonoine B

  • Takashi Nishiyama,
  • Erina Hamada,
  • Daishi Ishii,
  • Yuuto Kihara,
  • Nanase Choshi,
  • Natsumi Nakanishi,
  • Mari Murakami,
  • Kimiko Taninaka,
  • Noriyuki Hatae and
  • Tominari Choshi
Published 26 Jan 2021
Beilstein Arch. 2021, 20216. doi:10.3762/bxiv.2021.6.v1

Borylated methyl cinnamates: Expedited synthesis, characterization, crystallographic analysis and biological activities in glycosidase inhibition and in cancer cells lines.

  • William J Legge,
  • Yuna Shimadate,
  • Mahdi Ghorbani,
  • Jennette Sakoff,
  • Todd A Houston,
  • Atsushi Kato,
  • Paul Bernhardt and
  • Michela I. Simone
Published 22 Jan 2021
Beilstein Arch. 2021, 20214. doi:10.3762/bxiv.2021.4.v1

Metal-free visible-light-enabled vicinal trifluoromethyl dithiolation of unactivated alkenes

  • Xiaojuan Li,
  • Qiang Zhang,
  • Weigang Zhang,
  • Jinzhu Ma,
  • Yi Wang and
  • Yi Pan
Published 13 Jan 2021
Beilstein Arch. 2021, 20211. doi:10.3762/bxiv.2021.1.v1

β-Lactamase inhibition profile of new amidine substituted diazabicyclooctanes

  • zafar iqbal,
  • Yuanyu Gao,
  • Dong Tang,
  • Xueqin Ma,
  • Jinbo Ji,
  • Jian Sun,
  • Jingwen Ji,
  • Yuanbai Liu,
  • Lijuan Zhai,
  • Rui Jiang,
  • Yangxiu Mu,
  • Lili He,
  • Haikang Yang and
  • Zhixiang Yang
Published 21 Dec 2020
Beilstein Arch. 2020, 2020143. doi:10.3762/bxiv.2020.143.v1
Published 14 Dec 2020
Beilstein Arch. 2020, 2020142. doi:10.3762/bxiv.2020.142.v1
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