Correction: Mechanochemical enzymatic resolution of N-benzylated-β³-amino esters

• Mario Pérez-Venegas,
• Gloria Reyes-Rangel,
• Adrián Neri,
• Jaime Escalante and
• Eusebio Juaristi

Beilstein J. Org. Chem. 2017, 13, 2128–2130, doi:10.3762/bjoc.13.210

• Mario Perez-Venegas Gloria Reyes-Rangel Adrian Neri Jaime Escalante Eusebio Juaristi Departamento de Química, Centro de Investigación y de Estudios Avanzados, Avenida I.P.N. 2508, Ciudad de México, 07360, Mexico Centro de Investigaciones Químicas, Universidad Autónoma del Estado de Morelos, Av

Mechanically induced oxidation of alcohols to aldehydes and ketones in ambient air: Revisiting TEMPO-assisted oxidations

• Andrea Porcheddu,
• Evelina Colacino,
• Giancarlo Cravotto,
• Francesco Delogu and
• Lidia De Luca

Beilstein J. Org. Chem. 2017, 13, 2049–2055, doi:10.3762/bjoc.13.202

• ) UMR5247 CNRS-UM-ENSCM, Université de Montpellier, Place Eugène Bataillon, cc1703, 34095 Montpellier Cedex 05, France Dipartimento di Scienza e Tecnologia del Farmaco, University of Turin, Via P. Giuria, 9, 10125 Turin, Italy Dipartimento di Ingegneria Meccanica, Chimica e dei Materiali, Università degli

Influence of the milling parameters on the nucleophilic substitution reaction of activated β-cyclodextrins

• László Jicsinszky,
• Kata Tuza,
• Giancarlo Cravotto,
• Andrea Porcheddu,
• Francesco Delogu and
• Evelina Colacino

Beilstein J. Org. Chem. 2017, 13, 1893–1899, doi:10.3762/bjoc.13.184

• Laszlo Jicsinszky Kata Tuza Giancarlo Cravotto Andrea Porcheddu Francesco Delogu Evelina Colacino Dipartimento di Scienza e Tecnologia del Farmaco, University of Turin, via P. Giuria 9, 10125 Turin, Italy Cyclolab Cyclodextrin R&D Laboratory, Ltd., Illatos út 7, 1192 Budapest, Hungary Dipartimento

Mechanochemical enzymatic resolution of N-benzylated-β³-amino esters

• Mario Pérez-Venegas,
• Gloria Reyes-Rangel,
• Adrián Neri,
• Jaime Escalante and
• Eusebio Juaristi

Beilstein J. Org. Chem. 2017, 13, 1728–1734, doi:10.3762/bjoc.13.167

• Mario Perez-Venegas Gloria Reyes-Rangel Adrian Neri Jaime Escalante Eusebio Juaristi Departamento de Química, Centro de Investigación y de Estudios Avanzados, Avenida I.P.N. 2508, Ciudad de México, 07360, Mexico Centro de Investigaciones Químicas, Universidad Autónoma del Estado de Morelos, Av

An improved preparation of phorbol from croton oil

• Alberto Pagani,
• Simone Gaeta,
• Andrei I. Savchenko,
• Craig M. Williams and
• Giovanni Appendino

Beilstein J. Org. Chem. 2017, 13, 1361–1367, doi:10.3762/bjoc.13.133

• Alberto Pagani Simone Gaeta Andrei I. Savchenko Craig M. Williams Giovanni Appendino Dipartimento di Scienze del Farmaco, Università degli Studi del Piemonte Orientale, Largo Donegani 2, 28100 Novara, Italy School of Chemistry and Molecular Biosciences, University of Queensland, 4072, Brisbane

• EcoBiotics Ltd, QBiotics Ltd, the University of Queensland and the Università degli Studi del Piemonte Orientale for financial support, and Adipogen Life Sciences (San Diego, USA) for providing the samples of croton oil used in this investigation.

Continuous-flow processes for the catalytic partial hydrogenation reaction of alkynes

• Carmen Moreno-Marrodan,
• Francesca Liguori and
• Pierluigi Barbaro

Beilstein J. Org. Chem. 2017, 13, 734–754, doi:10.3762/bjoc.13.73

• Carmen Moreno-Marrodan Francesca Liguori Pierluigi Barbaro Consiglio Nazionale delle Ricerche, Istituto di Chimica dei Composti Organo Metallici, Via Madonna del Piano 10, 50019 Sesto Fiorentino, Firenze, Italy 10.3762/bjoc.13.73 Abstract The catalytic partial hydrogenation of substituted alkynes

Inclusion complexes of β-cyclodextrin with tricyclic drugs: an X-ray diffraction, NMR and molecular dynamics study

• Franca Castiglione,
• Fabio Ganazzoli,
• Luciana Malpezzi,
• Andrea Mele,
• Walter Panzeri and
• Giuseppina Raffaini

Beilstein J. Org. Chem. 2017, 13, 714–719, doi:10.3762/bjoc.13.70

• Franca Castiglione Fabio Ganazzoli Luciana Malpezzi Andrea Mele Walter Panzeri Giuseppina Raffaini Dipartimento di Chimica, Materiali e Ingegneria Chimica ‘G. Natta’, Politecnico di Milano, via Mancinelli 7, 20131 Milano, Italy CNR-Istituto di Chimica del Riconoscimento Molecolare – Via Mancinelli

Synthesis of spiro[isoindole-1,5’-isoxazolidin]-3(2H)-ones as potential inhibitors of the MDM2-p53 interaction

• Salvatore V. Giofrè,
• Santa Cirmi,
• Raffaella Mancuso,
• Francesco Nicolò,
• Giuseppe Lanza,
• Laura Legnani,
• Agata Campisi,
• Maria A. Chiacchio,
• Michele Navarra,
• Bartolo Gabriele and
• Roberto Romeo

Beilstein J. Org. Chem. 2016, 12, 2793–2807, doi:10.3762/bjoc.12.278

• Dipartimento di Chimica e Tecnologie Chimiche, Università della Calabria, Via P. Bucci, 12/C, 87036 Arcavacata di Rende (CS), Italy Dipartimento di Scienze Chimiche, Biologiche, Farmaceutiche e Ambientali, Università di Messina, Viale F. Stagno d'Alcontres 31, 98166 Messina, Italy Dipartimento di Scienze del

Towards the development of continuous, organocatalytic, and stereoselective reactions in deep eutectic solvents

• Davide Brenna,
• Elisabetta Massolo,
• Alessandra Puglisi,
• Sergio Rossi,
• Giuseppe Celentano,
• Maurizio Benaglia and
• Vito Capriati

Beilstein J. Org. Chem. 2016, 12, 2620–2626, doi:10.3762/bjoc.12.258

• Mangiagalli 25, 20133 Milano, Italy Dipartimento di Farmacia–Scienze del Farmaco, Università di Bari “Aldo Moro”, Consorzio C.I.N.M.P.I.S., Via E. Orabona 4, I-70125 Bari, Italy 10.3762/bjoc.12.258 Abstract Different deep eutectic solvent (DES) mixtures were studied as reaction media for the continuous

Useful access to enantiomerically pure protected inositols from carbohydrates: the aldohexos-5-uloses route

• Felicia D’Andrea,
• Giorgio Catelani,
• Lorenzo Guazzelli and
• Venerando Pistarà

Beilstein J. Org. Chem. 2016, 12, 2343–2350, doi:10.3762/bjoc.12.227

• Felicia D'Andrea Giorgio Catelani Lorenzo Guazzelli Venerando Pistara Università di Pisa, Dipartimento di Farmacia, Via Bonanno 33, 56126 Pisa, Italy Università di Catania, Dipartimento di Scienze del Farmaco, Viale A. Doria 6, 95125 Catania, Italy 10.3762/bjoc.12.227 Abstract The intramolecular

1H-Imidazol-4(5H)-ones and thiazol-4(5H)-ones as emerging pronucleophiles in asymmetric catalysis

• Antonia Mielgo and
• Claudio Palomo

Beilstein J. Org. Chem. 2016, 12, 918–936, doi:10.3762/bjoc.12.90

• Antonia Mielgo Claudio Palomo Departamento de Química Orgánica I, Facultad de Química, Universidad del País Vasco, Apdo. 1072, 20080 San Sebastián, Spain 10.3762/bjoc.12.90 Abstract Asymmetric catalysis represents a very powerful tool for the synthesis of enantiopure compounds. In this context

Interactions between 4-thiothymidine and water-soluble cyclodextrins: Evidence for supramolecular structures in aqueous solutions

• Vito Rizzi,
• Sergio Matera,
• Paola Semeraro,
• Paola Fini and
• Pinalysa Cosma

Beilstein J. Org. Chem. 2016, 12, 549–563, doi:10.3762/bjoc.12.54

• was supported by the COFIN-MIUR 2010 grant: “Architetture ibride multifunzionali basate su biomolecole per applicazioni nel campo della sensoristica, della conversione di energia e del biomedicale”. We gratefully acknowledge the skillful and excellent technical assistance of Mr. Sergio Nuzzo.

Enabling technologies and green processes in cyclodextrin chemistry

• Giancarlo Cravotto,
• Marina Caporaso,
• Laszlo Jicsinszky and
• Katia Martina

Beilstein J. Org. Chem. 2016, 12, 278–294, doi:10.3762/bjoc.12.30

• Giancarlo Cravotto Marina Caporaso Laszlo Jicsinszky Katia Martina Dipartimento di Scienza e Tecnologia del Farmaco and NIS - Centre for Nanostructured Interfaces and Surfaces, University of Turin, Via P. Giuria 9, 10125 Turin, Italy 10.3762/bjoc.12.30 Abstract The design of efficient synthetic

Investigation of the role of stereoelectronic effects in the conformation of piperidones by NMR spectroscopy and X-ray diffraction

• Cesar Garcias-Morales,
• David Ortegón-Reyna and
• Armando Ariza-Castolo

Beilstein J. Org. Chem. 2015, 11, 1973–1984, doi:10.3762/bjoc.11.213

• Cesar Garcias-Morales David Ortegon-Reyna Armando Ariza-Castolo Departamento de Química, Centro de Investigación y de Estudios Avanzados del Instituto Politécnico Nacional, Avenida Instituto Politécnico Nacional 2508 Colonia San Pedro Zacatenco, C.P. 07360, México, D.F., Mexico 10.3762/bjoc

Dicarboxylic esters: Useful tools for the biocatalyzed synthesis of hybrid compounds and polymers

• Ivan Bassanini,
• Karl Hult and
• Sergio Riva

Beilstein J. Org. Chem. 2015, 11, 1583–1595, doi:10.3762/bjoc.11.174

• Ivan Bassanini Karl Hult Sergio Riva Istituto di Chimica del Riconoscimento Molecolare, CNR, via Mario Bianco 9, Milano, Italy School of Biotechnology, Department of Industrial Biotechnology, Albanova KTH, Royal Institute of Technology, Stockholm, Sweden 10.3762/bjoc.11.174 Abstract Dicarboxylic

Tandem cross enyne metathesis (CEYM)–intramolecular Diels–Alder reaction (IMDAR). An easy entry to linear bicyclic scaffolds

• Javier Miró,
• María Sánchez-Roselló,
• Álvaro Sanz,
• Fernando Rabasa,
• Carlos del Pozo and
• Santos Fustero

Beilstein J. Org. Chem. 2015, 11, 1486–1493, doi:10.3762/bjoc.11.161

• Javier Miro Maria Sanchez-Rosello Alvaro Sanz Fernando Rabasa Carlos del Pozo Santos Fustero Departamento de Química Orgánica, Universidad de Valencia, E-46100 Burjassot, Spain Laboratorio de Moléculas Orgánicas, Centro de Investigación Príncipe Felipe, E-46012 Valencia, Spain 10.3762/bjoc.11.161

Highly selective palladium–benzothiazole carbene-catalyzed allylation of active methylene compounds under neutral conditions

• Antonio Monopoli,
• Pietro Cotugno,
• Carlo G. Zambonin,
• Francesco Ciminale and
• Angelo Nacci

Beilstein J. Org. Chem. 2015, 11, 994–999, doi:10.3762/bjoc.11.111

• Information File 250: General methods, synthetic procedures, characterization data of all new compounds. Acknowledgements We thank the University of Bari, the Italian Ministry of Instruction, University and Research (MIUR), and the Regione Puglia (“PON Ricerca e Competitività” 2007–2013—Avv. 254/Ric. del 18

Regulation of integrin and growth factor signaling in biomaterials for osteodifferentiation

• Qiang Wei,
• Theresa L. M. Pohl,
• Anja Seckinger,
• Joachim P. Spatz and
• Elisabetta A. Cavalcanti-Adam

Beilstein J. Org. Chem. 2015, 11, 773–783, doi:10.3762/bjoc.11.87

• regenerative medicine approaches. Reprinted with permission from [3]. Copyright 2011 Nature Publishing Group. (a) The structure of the integrin heterodimeric receptors with α and β subunits. (b) The major integrin–ligand combinations on the cell surfaces. Abbreviations: BSP, bone sialoprotein; Del-1

C-5’-Triazolyl-2’-oxa-3’-aza-4’a-carbanucleosides: Synthesis and biological evaluation

• Roberto Romeo,
• Caterina Carnovale,
• Salvatore V. Giofrè,
• Maria A. Chiacchio,
• Adriana Garozzo,
• Emanuele Amata,
• Giovanni Romeo and
• Ugo Chiacchio

Beilstein J. Org. Chem. 2015, 11, 328–334, doi:10.3762/bjoc.11.38

• Roberto Romeo Caterina Carnovale Salvatore V. Giofre Maria A. Chiacchio Adriana Garozzo Emanuele Amata Giovanni Romeo Ugo Chiacchio Dipartimento Scienze del Farmaco e dei Prodotti per la Salute, University of Messina, Via S.S. Annunziata, 98168 Messina, Italy Dipartimento di Scienze del Farmaco

Synthesis of modified cyclic and acyclic dextrins and comparison of their complexation ability

• Kata Tuza,
• László Jicsinszky,
• Tamás Sohajda,
• István Puskás and
• Éva Fenyvesi

Beilstein J. Org. Chem. 2014, 10, 2836–2843, doi:10.3762/bjoc.10.301

• Kata Tuza Laszlo Jicsinszky Tamas Sohajda Istvan Puskas Eva Fenyvesi CycloLab Cyclodextrin R&D Laboratory Ltd, Illatos út 7, Budapest, 1097, Hungary Dipartimento di Scienza e Tecnologia del Farmaco, Universitá di Torino, via P. Giuria 9, Turin, 10125, Italy 10.3762/bjoc.10.301 Abstract We

Synthesis and characterization of a hyper-branched water-soluble β-cyclodextrin polymer

• Francesco Trotta,
• Fabrizio Caldera,
• Roberta Cavalli,
• Andrea Mele,
• Carlo Punta,
• Lucio Melone,
• Franca Castiglione,
• Barbara Rossi,
• Monica Ferro,
• Vincenza Crupi,
• Domenico Majolino,
• Valentina Venuti and
• Dominique Scalarone

Beilstein J. Org. Chem. 2014, 10, 2586–2593, doi:10.3762/bjoc.10.271

• Dipartimento di Scienza e Tecnologia del Farmaco, Università di Torino, Via Pietro Giuria 9, 10125 Torino, Italy Department of Chemistry, Materials and Chemical Engineering “G. Natta”, Politecnico di Milano, Piazza L. da Vinci 32, 20132 Milano, Italy Elettra - Sincrotrone Trieste. Strada Statale 14 km 163.5

Phosphinocyclodextrins as confining units for catalytic metal centres. Applications to carbon–carbon bond forming reactions

• Matthieu Jouffroy,
• Rafael Gramage-Doria,
• David Sémeril,
• Dominique Armspach,
• Dominique Matt,
• Werner Oberhauser and
• Loïc Toupet

Beilstein J. Org. Chem. 2014, 10, 2388–2405, doi:10.3762/bjoc.10.249

• di Chimica dei Composti OrganoMetallici CNR, via Madonna del Piano, 10, 50019 Sesto Fiorentino, Firenze, Italy Groupe Matière Condensée et Matériaux, UMR 6626 CNRS, Université de Rennes 1, 263, avenue du Général Leclerc, 35042 Rennes Cedex, France 10.3762/bjoc.10.249 Abstract The capacity of two

Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration

• Michele Mari,
• Simone Lucarini,
• Francesca Bartoccini,
• Giovanni Piersanti and
• Gilberto Spadoni

Beilstein J. Org. Chem. 2014, 10, 1991–1998, doi:10.3762/bjoc.10.207

• Michele Mari Simone Lucarini Francesca Bartoccini Giovanni Piersanti Gilberto Spadoni Department of Biomolecular Sciences, University of Urbino “Carlo Bo”, Piazza del Rinascimento 6, 61029 Urbino (PU), Italy 10.3762/bjoc.10.207 Abstract The reaction of 3-substituted indoles with dehydroalanine

An experimental and theoretical NMR study of NH-benzimidazoles in solution and in the solid state: proton transfer and tautomerism

• Carla I. Nieto,
• Pilar Cabildo,
• M. Ángeles García,
• Rosa M. Claramunt,
• Ibon Alkorta and
• José Elguero

Beilstein J. Org. Chem. 2014, 10, 1620–1629, doi:10.3762/bjoc.10.168

• Carla I. Nieto Pilar Cabildo M. Angeles Garcia Rosa M. Claramunt Ibon Alkorta Jose Elguero Departamento de Química Orgánica y Bio-Orgánica, Facultad de Ciencias, UNED Senda del Rey 9, E-28040 Madrid, Spain Instituto de Química Médica, CSIC, Juan de la Cierva, 3, E-28006 Madrid, Spain 10.3762/bjoc

Pd/C-catalyzed aerobic oxidative esterification of alcohols and aldehydes: a highly efficient microwave-assisted green protocol

• Marina Caporaso,
• Giancarlo Cravotto,
• Spyros Georgakopoulos,
• George Heropoulos,
• Katia Martina and
• Silvia Tagliapietra

Beilstein J. Org. Chem. 2014, 10, 1454–1461, doi:10.3762/bjoc.10.149

• Marina Caporaso Giancarlo Cravotto Spyros Georgakopoulos George Heropoulos Katia Martina Silvia Tagliapietra Dipartimento di Scienza e Tecnologia del Farmaco, University of Turin, Via P. Giuria 9, 10125 Torino, Italy. Fax +390116707687; Tel: +390116707684 Interdepartmental Centre “Nanostructured